6ONI-D-B

PDB Title CRYSTAL STRUCTURE OF PPARGAMMA LIGAND BINDING DOMAIN IN COMPLEX WITH N-COR PEPTIDE AND INVERSE AGONIST T0070907
Resolution (Å) 1.800
Classification TRANSCRIPTION/AGONIST

Protein

Description Peroxisome proliferator-activated receptor gamma
Organism Homo sapiens
Chain B
Length 262
Binding Area (Å2) 479.58
Molecular Weight -
Aromaticity 0.08
Instability -
Isoelectric Point 5.34
Sequence QLNPESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDLYX

Peptide

Description NCOR isoform c
Organism Homo sapiens
Chain D
Length 13
Binding Area (Å2) 570.75
Hydrophobic (% a.a.)
61%
Molecular Weight 1485.79
Aromaticity 0.00
Instability 24.05
Isoelectric Point 6.07
Sequence NLGLEDIIRKALM

Clustering Classification

Sequence cluster S 198
Contact cluster C8
Interface cluster I1734