PDB Title | CRYSTAL STRUCTURE OF THE ER-ALPHA LIGAND-BINDING DOMAIN (Y537S) IN COMPLEX WITH THE PHENYLAMINO-SUBSTITUTED ESTROGEN, (8R,9S,13S,14S, 17S)-13-METHYL-17-(PHENYLAMINO)-7,8,9,11,12,13,14,15,16,17-DECAHYDRO- 6H-CYCLOPENTA[A]PHENANTHREN-3-OL |
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Resolution (Å) | 2.380 |
Classification | TRANSCRIPTION |
Description | Estrogen receptor |
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Organism | Homo sapiens |
Chain | B |
Length | 236 |
Binding Area (Å2) | 466.64 |
Molecular Weight | - |
Aromaticity | 0.05 |
Instability | - |
Isoelectric Point | 5.92 |
Sequence | SLALSLTADQMVSALLDAEPPILYSEYDPTRPSEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLECAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKCVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMKCKVVPLSDLLLEMLDAHRX |
Description | NUCLEAR RECEPTOR COACTIVATOR 2 |
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Organism | Homo sapiens |
Chain | D |
Length | 9 |
Binding Area (Å2) | 526.17 |
Hydrophobic (% a.a.) |
|
Molecular Weight | 1135.36 |
Aromaticity | 0.00 |
Instability | 78.48 |
Isoelectric Point | 8.76 |
Sequence | KILHRLLQD |
Is the complex classified in the same cluster?