1T5Z-B-A

PDB Title CRYSTAL STRUCTURE OF THE ANDROGEN RECEPTOR LIGAND BINDING DOMAIN (LBD) WITH DHT AND A PEPTIDE DERIVED FROM ITS PHYSIOLOGICAL COACTIVATOR ARA70
Resolution (Å) 2.300
Classification HORMONE/GROWTH FACTOR

Protein

Description Androgen receptor
Organism Homo sapiens
Chain A
Length 251
Binding Area (Å2) 548.04
Molecular Weight -
Aromaticity 0.11
Instability -
Isoelectric Point 8.88
Sequence CQPIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIACKRKNPTSCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHTX

Peptide

Description Nuclear receptor coactivator 4
Organism Homo sapiens
Chain B
Length 11
Binding Area (Å2) 612.85
Hydrophobic (% a.a.)
36%
Molecular Weight 1389.59
Aromaticity 0.27
Instability 45.16
Isoelectric Point 8.22
Sequence SEKFKLLFQSY

Clustering Classification

Sequence cluster S 916
Contact cluster C9
Interface cluster I5