4OFU-B-A

PDB Title CRYSTAL STRUCTURE OF AR-LBD BOUND WITH CO-REGULATOR PEPTIDE
Resolution (Å) 2.120
Classification HORMONE RECEPTOR/PEPTIDE

Protein

Description Androgen receptor
Organism Homo sapiens
Chain A
Length 242
Binding Area (Å2) 424.97
Molecular Weight -
Aromaticity 0.12
Instability -
Isoelectric Point 8.11
Sequence PIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSAMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIASCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHTX

Peptide

Description co-regulator peptide
Organism synthetic construct
Chain B
Length 8
Binding Area (Å2) 538.84
Hydrophobic (% a.a.)
25%
Molecular Weight 994.06
Aromaticity 0.38
Instability 28.21
Isoelectric Point 8.31
Sequence SAFSRYYT

Clustering Classification

Sequence cluster S 496
Contact cluster C9
Interface cluster I5