4OKW-B-A

PDB Title CRYSTAL STRUCTURE OF W741L-AR-LBD BOUND WITH CO-REGULATOR PEPTIDE
Resolution (Å) 2.000
Classification HORMONE RECEPTOR/PEPTIDE

Protein

Description Androgen receptor
Organism Homo sapiens
Chain A
Length 240
Binding Area (Å2) 407.74
Molecular Weight -
Aromaticity 0.11
Instability -
Isoelectric Point 8.11
Sequence PIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSLMGLMVFAMGWRSFTNVNSAMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIACSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHX

Peptide

Description co-regulator peptide
Organism -
Chain B
Length 8
Binding Area (Å2) 512.82
Hydrophobic (% a.a.)
25%
Molecular Weight 1010.06
Aromaticity 0.25
Instability 68.96
Isoelectric Point 5.08
Sequence DTLFSQHY

Clustering Classification

Sequence cluster S 1452
Contact cluster C9
Interface cluster I5