4OKX-B-A

PDB Title CRYSTAL STRUCTURE OF W741L-AR-LBD BOUND WITH CO-REGULATOR PEPTIDE
Resolution (Å) 2.100
Classification HORMONE RECEPTOR/PEPTIDE

Protein

Description Androgen receptor
Organism Homo sapiens
Chain A
Length 241
Binding Area (Å2) 367.77
Molecular Weight -
Aromaticity 0.11
Instability -
Isoelectric Point 8.11
Sequence PIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSLMGLMVFAMGWRSFTNVNSAMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIACSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHTX

Peptide

Description co-regulator peptide
Organism -
Chain B
Length 8
Binding Area (Å2) 457.54
Hydrophobic (% a.a.)
12%
Molecular Weight 1061.10
Aromaticity 0.38
Instability -1.86
Isoelectric Point 5.55
Sequence SFRDWYTS

Clustering Classification

Sequence cluster S 538
Contact cluster C9
Interface cluster I5