2Q7K-B-A

PDB Title THE ANDROGEN RECEPTOR PROSTATE CANCER MUTANT H874Y LIGAND BINDING DOMAIN BOUND WITH TESTOSTERONE AND AN AR 20-30 PEPTIDE
Resolution (Å) 1.800
Classification HORMONE

Protein

Description Androgen receptor
Organism Homo sapiens
Chain A
Length 243
Binding Area (Å2) 463.31
Molecular Weight -
Aromaticity 0.12
Instability -
Isoelectric Point 8.46
Sequence PIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIASCSRRFYQLTKLLDSVQPIARELYQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHTQX

Peptide

Description Androgen receptor
Organism Homo sapiens
Chain B
Length 10
Binding Area (Å2) 550.89
Hydrophobic (% a.a.)
60%
Molecular Weight 1110.22
Aromaticity 0.20
Instability 44.45
Isoelectric Point 5.52
Sequence GAFQNLFQSV

Clustering Classification

Sequence cluster S 223
Contact cluster C9
Interface cluster I5