4OEZ-B-A

PDB Title CRYSTAL STRUCTURE OF AR-LBD BOUND WITH CO-REGULATOR PEPTIDE
Resolution (Å) 1.800
Classification HORMONE RECEPTOR/PEPTIDE

Protein

Description Androgen receptor
Organism Homo sapiens
Chain A
Length 243
Binding Area (Å2) 410.66
Molecular Weight -
Aromaticity 0.12
Instability -
Isoelectric Point 7.86
Sequence QPIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSAMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIASCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHTX

Peptide

Description co-regulator peptide
Organism synthetic construct
Chain B
Length 8
Binding Area (Å2) 521.31
Hydrophobic (% a.a.)
37%
Molecular Weight 944.04
Aromaticity 0.25
Instability 22.21
Isoelectric Point 8.46
Sequence SAFSRLYT

Clustering Classification

Sequence cluster S 496
Contact cluster C9
Interface cluster I5