4OEY-B-A

PDB Title CRYSTAL STRUCTURE OF AR-LBD BOUND WITH CO-REGULATOR PEPTIDE
Resolution (Å) 1.830
Classification HORMONE RECEPTOR/PEPTIDE

Protein

Description Androgen receptor
Organism Homo sapiens
Chain A
Length 242
Binding Area (Å2) 403.95
Molecular Weight -
Aromaticity 0.12
Instability -
Isoelectric Point 8.11
Sequence PIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSAMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIASCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHTX

Peptide

Description co-regulator peptide
Organism synthetic construct
Chain B
Length 8
Binding Area (Å2) 523.15
Hydrophobic (% a.a.)
62%
Molecular Weight 924.01
Aromaticity 0.25
Instability -1.86
Isoelectric Point 5.52
Sequence GAFQNLFQ

Clustering Classification

Sequence cluster S 223
Contact cluster C9
Interface cluster I5