4OHA-B-A

PDB Title CRYSTAL STRUCTURE OF T877A-AR-LBD BOUND WITH CO-REGULATOR PEPTIDE
Resolution (Å) 1.420
Classification HORMONE RECEPTOR/PEPTIDE

Protein

Description Androgen receptor
Organism Homo sapiens
Chain A
Length 243
Binding Area (Å2) 390.38
Molecular Weight -
Aromaticity 0.12
Instability -
Isoelectric Point 8.11
Sequence PIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSAMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIASCSRRFYQLTKLLDSVQPIARELHQFAFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHTQX

Peptide

Description co-regulator peptide
Organism -
Chain B
Length 9
Binding Area (Å2) 503.23
Hydrophobic (% a.a.)
33%
Molecular Weight 1100.23
Aromaticity 0.22
Instability 20.86
Isoelectric Point 10.83
Sequence SAFSRLYTR

Clustering Classification

Sequence cluster S 496
Contact cluster C9
Interface cluster I5