3V4A-B-A

PDB Title STRUCTURE OF AR LBD WITH ACTIVATOR PEPTIDE AND SARM INHIBITOR 2
Resolution (Å) 1.950
Classification TRANSCRIPTION

Protein

Description Androgen receptor
Organism Homo sapiens
Chain A
Length 245
Binding Area (Å2) 495.00
Molecular Weight -
Aromaticity 0.11
Instability -
Isoelectric Point 8.41
Sequence PIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIACTSCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHTQX

Peptide

Description Androgen receptor
Organism Homo sapiens
Chain B
Length 11
Binding Area (Å2) 590.03
Hydrophobic (% a.a.)
54%
Molecular Weight 1266.40
Aromaticity 0.18
Instability 41.32
Isoelectric Point 9.75
Sequence GAFQNLFQSVR

Clustering Classification

Sequence cluster S 223
Contact cluster C9
Interface cluster I5