4OKT-B-A

PDB Title CRYSTAL STRUCTURE OF W741L-AR-LBD BOUND WITH CO-REGULATOR PEPTIDE
Resolution (Å) 2.500
Classification HORMONE RECEPTOR/PEPTIDE

Protein

Description Androgen receptor
Organism Homo sapiens
Chain A
Length 249
Binding Area (Å2) 494.60
Molecular Weight -
Aromaticity 0.11
Instability -
Isoelectric Point 8.85
Sequence QPIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSLMGLMVFAMGWRSFTNVNSAMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIAKRKNPTSCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHTX

Peptide

Description co-regulator peptide
Organism -
Chain B
Length 11
Binding Area (Å2) 594.29
Hydrophobic (% a.a.)
27%
Molecular Weight 1302.39
Aromaticity 0.18
Instability 76.34
Isoelectric Point 8.75
Sequence DSAFSRLYTRS

Clustering Classification

Sequence cluster S 496
Contact cluster C9
Interface cluster I5