4OH5-B-A

PDB Title CRYSTAL STRUCTURE OF T877A-AR-LBD BOUND WITH CO-REGULATOR PEPTIDE
Resolution (Å) 2.000
Classification HORMONE RECEPTOR/PEPTIDE

Protein

Description Androgen receptor
Organism Homo sapiens
Chain A
Length 243
Binding Area (Å2) 389.21
Molecular Weight -
Aromaticity 0.12
Instability -
Isoelectric Point 8.11
Sequence PIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSAMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIASCSRRFYQLTKLLDSVQPIARELHQFAFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHTQX

Peptide

Description co-regulator peptide
Organism -
Chain B
Length 9
Binding Area (Å2) 492.37
Hydrophobic (% a.a.)
55%
Molecular Weight 1011.09
Aromaticity 0.22
Instability 48.28
Isoelectric Point 5.52
Sequence GAFQNLFQS

Clustering Classification

Sequence cluster S 223
Contact cluster C9
Interface cluster I5