4OFR-B-A

PDB Title CRYSTAL STRUCTURE OF AR-LBD BOUND WITH CO-REGULATOR PEPTIDE
Resolution (Å) 2.260
Classification HORMONE RECEPTOR/PEPTIDE

Protein

Description Androgen receptor
Organism Homo sapiens
Chain A
Length 244
Binding Area (Å2) 502.27
Molecular Weight -
Aromaticity 0.11
Instability -
Isoelectric Point 8.11
Sequence PIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSAMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIAPTSCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHTX

Peptide

Description co-regulator peptide
Organism synthetic construct
Chain B
Length 8
Binding Area (Å2) 578.02
Hydrophobic (% a.a.)
12%
Molecular Weight 1061.10
Aromaticity 0.38
Instability 22.21
Isoelectric Point 5.55
Sequence SSFRDWYT

Clustering Classification

Sequence cluster S 538
Contact cluster C9
Interface cluster I5