4LSJ-B-A

PDB Title CRYSTAL STRUCTURE OF THE GLUCOCORTICOID RECEPTOR LIGAND BINDING DOMAIN BOUND TO A DIBENZOXAPINE SULFONAMIDE
Resolution (Å) 2.350
Classification TRANSCRIPTION

Protein

Description Glucocorticoid receptor
Organism Homo sapiens
Chain A
Length 246
Binding Area (Å2) 495.35
Molecular Weight -
Aromaticity 0.11
Instability -
Isoelectric Point 6.26
Sequence PQLTPTLVSLLEVIEPEVLYAGYDSSVPDSTWRIMTTLNMLGGRQVIAAVKWAKAIPGFRNLHLDDQMTLLQYSWMYLMAFALGWRSYRQSSANLLCFAPDLIINEQRMTLPGMYDQCKHMLYVSSELHRLQVSYEEYLCMKTLLLLSSVPKDGLKSQELFDEIRMTYIKELGKAIVNWQRFYQLTKLLDSMHEVVENLLNYCFQTFLDKTMSIEFPEMLAEIITNQIPKYSNGNIKKLLFHQKXX

Peptide

Description D30 peptide
Organism -
Chain B
Length 10
Binding Area (Å2) 609.08
Hydrophobic (% a.a.)
40%
Molecular Weight 1263.46
Aromaticity 0.10
Instability 71.20
Isoelectric Point 4.85
Sequence SSRLWELLME

Clustering Classification

Sequence cluster S 130
Contact cluster C9
Interface cluster I1253