2PKL-B-A

PDB Title ANDROGEN RECEPTOR LBD WITH SMALL MOLECULE
Resolution (Å) 2.490
Classification HORMONE RECEPTOR

Protein

Description Androgen receptor
Organism Homo sapiens
Chain A
Length 251
Binding Area (Å2) 306.43
Molecular Weight -
Aromaticity 0.11
Instability -
Isoelectric Point 8.94
Sequence QPIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIACKRKNPTSCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHTXX

Peptide

Description ARA70 peptide
Organism -
Chain B
Length 4
Binding Area (Å2) 372.90
Hydrophobic (% a.a.)
75%
Molecular Weight 519.68
Aromaticity 0.25
Instability -13.73
Isoelectric Point 8.75
Sequence KLLF

Clustering Classification

Sequence cluster S 1130
Contact cluster C1009
Interface cluster I5