6PDI-B-A

PDB Title HUMAN PIM1 BOUND TO BENZOTHIOPHENE INHIBITOR 224
Resolution (Å) 1.850
Classification TRANSFERASE/TRANSFERASE INHIBITOR

Protein

Description Serine/threonine-protein kinase pim-1
Organism Homo sapiens
Chain A
Length 275
Binding Area (Å2) 501.85
Molecular Weight -
Aromaticity 0.10
Instability -
Isoelectric Point 5.14
Sequence EPLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIGGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHX

Peptide

Description Peptide
Organism synthetic construct
Chain B
Length 10
Binding Area (Å2) 654.67
Hydrophobic (% a.a.)
30%
Molecular Weight 1220.39
Aromaticity 0.00
Instability 191.80
Isoelectric Point 12.48
Sequence ARKRRRHPSG

Clustering Classification

Sequence cluster S 217
Contact cluster C17
Interface cluster I17