5MZL-B-A

PDB Title CRYSTAL STRUCTURE OF HUMAN PIM-1 KINASE IN COMPLEX WITH A CONSENSUSPEPTIDE AND FRAGMENT LIKE MOLEKULE N-QUINOLIN-5-YLPYRIDINE- 3-CARBOXAMIDE
Resolution (Å) 1.960
Classification TRANSFERASE

Protein

Description Serine/threonine-protein kinase pim-1
Organism Homo sapiens
Chain A
Length 270
Binding Area (Å2) 452.63
Molecular Weight -
Aromaticity 0.10
Instability -
Isoelectric Point 5.20
Sequence PLESQYQVGPLLGSSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIGGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHX

Peptide

Description Pimtide
Organism Homo sapiens
Chain B
Length 8
Binding Area (Å2) 608.87
Hydrophobic (% a.a.)
12%
Molecular Weight 1092.26
Aromaticity 0.00
Instability 237.25
Isoelectric Point 12.48
Sequence RKRRRHPS

Clustering Classification

Sequence cluster S 217
Contact cluster C17
Interface cluster I17