5N5L-B-A

PDB Title CRYSTAL STRUCTURE OF HUMAN PIM-1 KINASE IN COMPLEX WITH A CONSENSUSPEPTIDE AND [2-OXO-2-(1H-PYRROL-2-YL)ETHYL] 5-BROMO-1H- INDOLE-3-CARBOXYLATE
Resolution (Å) 1.970
Classification TRANSFERASE

Protein

Description Serine/threonine-protein kinase pim-1
Organism Homo sapiens
Chain A
Length 273
Binding Area (Å2) 517.03
Molecular Weight -
Aromaticity 0.10
Instability -
Isoelectric Point 5.20
Sequence PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIGGQVFFRQRVSXECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHX

Peptide

Description Pimtide
Organism Homo sapiens
Chain B
Length 9
Binding Area (Å2) 675.85
Hydrophobic (% a.a.)
22%
Molecular Weight 1149.31
Aromaticity 0.00
Instability 212.00
Isoelectric Point 12.48
Sequence RKRRRHPSG

Clustering Classification

Sequence cluster S 217
Contact cluster C17
Interface cluster I17