4GW8-B-A

PDB Title HUMAN PROTO-ONCOGENE SERINE THREONINE KINASE (PIM1) IN COMPLEX WITH A CONSENSUS PEPTIDE AND LEUCETTINE L41
Resolution (Å) 2.000
Classification TRANSFERASE

Protein

Description Serine/threonine-protein kinase pim-1
Organism Homo sapiens
Chain A
Length 274
Binding Area (Å2) 516.44
Molecular Weight -
Aromaticity 0.10
Instability -
Isoelectric Point 5.20
Sequence PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIGGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHX

Peptide

Description Consensus peptide (Pimtide)
Organism -
Chain B
Length 9
Binding Area (Å2) 668.52
Hydrophobic (% a.a.)
22%
Molecular Weight 1149.31
Aromaticity 0.00
Instability 212.00
Isoelectric Point 12.48
Sequence RKRRRHPSG

Clustering Classification

Sequence cluster S 217
Contact cluster C17
Interface cluster I17