2BZK-A-B

PDB Title CRYSTAL STRUCTURE OF THE HUMAN PIM1 IN COMPLEX WITH AMPPNP AND PIMTIDE
Resolution (Å) 2.450
Classification TRANSFERASE/PEPTIDE

Protein

Description PROTO-ONCOGENE SERINE THREONINE PROTEIN KINASE PIM1
Organism Homo sapiens
Chain B
Length 269
Binding Area (Å2) 420.23
Molecular Weight -
Aromaticity 0.10
Instability -
Isoelectric Point 5.20
Sequence PLESQYQVGPLLGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIGGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHX

Peptide

Description PIMTIDE
Organism Homo sapiens
Chain A
Length 7
Binding Area (Å2) 546.64
Hydrophobic (% a.a.)
14%
Molecular Weight 936.08
Aromaticity 0.00
Instability 269.71
Isoelectric Point 12.30
Sequence KRRRHPS

Clustering Classification

Sequence cluster S 217
Contact cluster C17
Interface cluster I17