2C3I-A-B

PDB Title CRYSTAL STRUCTURE OF HUMAN PIM1 IN COMPLEX WITH IMIDAZOPYRIDAZIN I
Resolution (Å) 1.900
Classification TRANSFERASE/PEPTIDE

Protein

Description PROTO-ONCOGENE SERINE THREONINE PROTEIN KINASE PIM1
Organism Homo sapiens
Chain B
Length 267
Binding Area (Å2) 481.32
Molecular Weight -
Aromaticity 0.10
Instability -
Isoelectric Point 5.28
Sequence QYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGEGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIGGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHX

Peptide

Description PIMTIDE
Organism Homo sapiens
Chain A
Length 8
Binding Area (Å2) 617.95
Hydrophobic (% a.a.)
25%
Molecular Weight 993.13
Aromaticity 0.00
Instability 237.25
Isoelectric Point 12.30
Sequence KRRRHPSG

Clustering Classification

Sequence cluster S 217
Contact cluster C17
Interface cluster I17