3MA3-B-A

PDB Title CRYSTAL STRUCTURE OF HUMAN PROTO-ONCOGENE SERINE THREONINE KINASE (PIM1) IN COMPLEX WITH A CONSENSUS PEPTIDE AND A NAPHTHO-DIFURAN LIGAND
Resolution (Å) 2.300
Classification TRANSFERASE

Protein

Description Proto-oncogene serine/threonine-protein kinase pim-1
Organism Homo sapiens
Chain A
Length 268
Binding Area (Å2) 412.87
Molecular Weight -
Aromaticity 0.10
Instability -
Isoelectric Point 5.28
Sequence QYQVGPLLGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIGGQVFFRQRVSXECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHX

Peptide

Description Pimtide
Organism -
Chain B
Length 7
Binding Area (Å2) 554.69
Hydrophobic (% a.a.)
14%
Molecular Weight 936.08
Aromaticity 0.00
Instability 269.71
Isoelectric Point 12.30
Sequence KRRRHPS

Clustering Classification

Sequence cluster S 217
Contact cluster C17
Interface cluster I17