3CY2-B-A

PDB Title CRYSTAL STRUCTURE OF HUMAN PROTO-ONCOGENE SERINE THREONINE KINASE (PIM1) IN COMPLEX WITH A CONSENSUS PEPTIDE AND A BETA CARBOLINE LIGAND II
Resolution (Å) 2.010
Classification TRANSFERASE

Protein

Description Proto-oncogene serine/threonine-protein kinase Pim-1, Isoform 2
Organism Homo sapiens
Chain A
Length 273
Binding Area (Å2) 485.20
Molecular Weight -
Aromaticity 0.10
Instability -
Isoelectric Point 5.20
Sequence PLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIGGQVFFRQRVSSECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHXX

Peptide

Description Pimtide peptide
Organism -
Chain B
Length 9
Binding Area (Å2) 634.43
Hydrophobic (% a.a.)
22%
Molecular Weight 1149.31
Aromaticity 0.00
Instability 212.00
Isoelectric Point 12.48
Sequence RKRRRHPSG

Clustering Classification

Sequence cluster S 217
Contact cluster C17
Interface cluster I17