5CJ6-B-A

PDB Title CRYSTAL STRUCTURE OF A SELECTIVE ANDROGEN RECEPTOR MODULATOR BOUND TO THE LIGAND BINDING DOMAIN OF THE HUMAN ANDROGEN RECEPTOR
Resolution (Å) 2.070
Classification SIGNALING PROTEIN

Protein

Description Androgen receptor
Organism Homo sapiens
Chain A
Length 245
Binding Area (Å2) 434.51
Molecular Weight -
Aromaticity 0.11
Instability -
Isoelectric Point 8.41
Sequence PIFLNVLEAIEPGVVCAGHDNNQPDSFAALLSSLNELGERQLVHVVKWAKALPGFRNLHVDDQMAVIQYSWMGLMVFAMGWRSFTNVNSRMLYFAPDLVFNEYRMHKSRMYSQCVRMRHLSQEFGWLQITPQEFLCMKALLLFSIIPVDGLKNQKFFDELRMNYIKELDRIIACPTSCSRRFYQLTKLLDSVQPIARELHQFTFDLLIKSHMVSVDFPEMMAEIISVQVPKILSGKVKPIYFHTX

Peptide

Description small peptide
Organism synthetic construct
Chain B
Length 10
Binding Area (Å2) 524.55
Hydrophobic (% a.a.)
60%
Molecular Weight 1110.22
Aromaticity 0.20
Instability 44.45
Isoelectric Point 5.52
Sequence GAFQNLFQSV

Clustering Classification

Sequence cluster S 223
Contact cluster C7
Interface cluster I5